Search results:


General Information



Gene_Symbol Gene_ID Gene_Name Chromosome Alias
ABCG2 9429 ATP-binding cassette, sub-family G (WHITE), member 2 (Junior blood group)  4EST157481, MXR, BCRP, ABCP, CD338 







  • Evidence
  • Gene
  • mRNA
  • CDS
  • Protein
  • PTM
  • Enzyme
  • PPi
  • Pathway
  • Structural
  • Domain
  • Ontology
  • SNP
  • Drug
  • External Links



Evidence Information


Pubmed ID Year Sample Information Techniques Mechanism Fold Change Remark
25793771   2015Cell line : -

Source : -

Sample Type : CRC Tumor

No. of Sample : -

Stage : -

real time RT-PCR,GenotypingDown-regulation-ABCG2 mRNA levels were significantly lower in adenomas and carcinomas compared to the level in unaffected tissue from the same individuals and compared to tissue from healthy individuals .

25427584   2014Cell line : -

Source : Telemark Hospital (Skien) and Oslo University Hospital (Oslo).

Sample Type : CRC Tumor

No. of Sample : -

Stage : -

Fluorescence activated cell sorting,,immunofluorescence, real-timeRT-PCR, multidrug resistance, and sphere formation assays Up-regulation-overexpression of ABCG2 and the expression of stem cell surface markers are collectively responsible for chemotherapy failure, tumor recurrence, and invasion in colon cancer.

25928015   2015Cell line : HCT8, HCT116, SW620 NSCLC, A549, NCI-H460

Source : ATCC

Sample Type : -

No. of Sample : -

Stage : -

Immunoblotting,Cell proliferation,viability assayUp-regulation--


Gene Details



NC_000004.11 (89011416..89152569, complement)

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Gene Type protein coding
Gene Family CD molecules, "ATP binding cassette transporters / subfamily G"
Description The membrane-associated protein encoded by this gene is included in the superfamily of ATP-binding cassette (ABC) transporters. ABC proteins transport various molecules across extra- and intra-cellular membranes. ABC genes are divided into seven distinct subfamilies (ABC1, MDR/TAP, MRP, ALD, OABP, GCN20, White). This protein is a member of the White subfamily. Alternatively referred to as a breast cancer resistance protein, this protein functions as a xenobiotic transporter which may play a major role in multi-drug resistance. It likely serves as a cellular defense mechanism in response to mitoxantrone and anthracycline exposure. Significant expression of this protein has been observed in the placenta, which may suggest a potential role for this molecule in placenta tissue. Multiple transcript variants encoding different isoforms have been found for this gene. [provided by RefSeq, Apr 2012]  
Chromosome 4
Location 4q22.1
Start 89011416  
End 89152569  
Strand -  
Gene Sequence

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Length 141154  
OMIM ID 603756   
HGNC ID HGNC:74   
Unigene ID Hs.480218   
Ensembl ID ENSG00000118777   
PharmGKB ID PA390   

mRNA Information


mRNA ID ?NM_001257386.1
Exon  
mRNA Sequence

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Length  



CDS Information


   
Location
CDS Sequence

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CCDS ID CCDS3628.1



Protein Information


      
Protein IDNP_001244315.1
Protein NameATP-binding cassette, sub-family G (WHITE), member 2 (Junior blood group)
Molecular Wt. (Da)0
Protein Sequence

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Length 655  
Uniprot IDQ9Y6Y1
Ensembl Protein ID ENSP00000306522  



Post-translational Modification Information (Source : HPRD)


Residue Type site
NGlycosylation596
SPhosphorylation100
SPhosphorylation103
SPhosphorylation2
SPhosphorylation65

Enzyme Information


No matching records could be found.

PPi Information


(Click to view network : Source STRING)      View   

No matching records from HPRD source could be found.

Pathway Information


            
Pathway Name Pathway ID
ABC transporters hsa02010
Bile secretion hsa04976


Structure Information


No matching records could be found.

Domain Information




ID Location Description
cd0321334-268  ABCG_EPDR
cl2145534-268  P-loop_NTPase superfamily
cd0323455-268  ABCG_White
cd0323234-262  ABCG_PDR_domain2
cd0323352-268  ABCG_PDR_domain1
pfam01061375-586  ABC2_membrane
cl21474375-586  ABC2_membrane superfamily
cd0326377-272  ABC_subfamily_A
cd0326461-268  ABC_drug_resistance_like
cd0322560-263  ABC_cobalt_CbiO_domain1
cd0325559-264  ABC_MJ0796_LolCDE_FtsE
cd0323061-264  ABC_DR_subfamily_A
pfam0000564-214  ABC_tran
cd0326672-268  ABC_NatA_sodium_exporter
cd0323561-268  ABC_Metallic_Cations
cd0326160-272  ABC_Org_Solvent_Resistant
cd0325960-268  ABC_Carb_Solutes_like
cd0321964-272  ABC_Mj1267_LivG_branched
cd0329337-243  ABC_NrtD_SsuB_transporters
cd0326860-268  ABC_BcrA_bacitracin_resist
cd0322960-263  ABC_Class3
cd0326577-272  ABC_DrrA
cd0026760-263  ABC_ATPase
cd0321460-268  ABC_Iron-Siderophores_B12_Hemin
cd0329774-268  ABC_ModC_molybdenum_transporter
cd0324557-264  ABCC_bacteriocin_exporters
cd0329264-243  ABC_FtsE_transporter
cd0322837-263  ABCC_MRP_Like
cd0329977-274  ABC_ModC_like
cd0325661-272  ABC_PhnC_transporter
cd0325360-274  ABCC_ATM1_transporter
cd0325736-240  ABC_NikE_OppD_transporters
cd0329877-268  ABC_ThiQ_thiamine_transporter
cd0322661-262  ABC_cobalt_CbiO_domain2
cd0326744-268  ABC_NatA_like
cd0324760-268  ABCC_cytochrome_bd
cd0324660-264  ABCC_Protease_Secretion
cd0325460-274  ABCC_Glucan_exporter_like
cd0322477-274  ABC_TM1139_LivF_branched
cd0326060-272  ABC_PstB_phosphate_transporter
cd0325257-274  ABCC_Hemolysin
cd0330178-243  ABC_MalK_N
cd0326260-244  ABC_HisP_GlnQ
cd0325862-272  ABC_MetN_methionine_transporter
cd0321877-272  ABC_YhbG
cd0326977-268  ABC_putative_ATPase
cd0325160-276  ABCC_MsbA
cd0330059-243  ABC_PotA_N
cd0323178-245  ABC_CcmA_heme_exporter
cd0329664-294  ABC_CysA_sulfate_importer
TIGR0118977-246  ccmA
cd0322038-268  ABC_KpsT_Wzt
cd0329564-264  ABC_OpuCA_Osmoprotection
cd0321760-282  ABC_FeS_Assembly
cd0325063-263  ABCC_MRP_domain1
cd0324960-243  ABC_MTABC3_MDL1_MDL2
cd0329478-297  ABC_Pro_Gly_Betaine
cd0324863-264  ABCC_TAP
cd0321677-264  ABC_Carb_Monos_I
cd0321577-240  ABC_Carb_Monos_II
cd0329064-247  ABCC_SUR1_N
cd0323778-230  ABC_RNaseL_inhibitor_domain2
cd0324437-243  ABCC_MRP_domain2
cd0322766-245  ABC_Class2
cd0322363-254  ABCD_peroxisomal_ALDP
cd0323678-243  ABC_RNaseL_inhibitor_domain1
cd0327945-245  ABC_sbcCD
cd0322160-217  ABCF_EF-3
cd0324073-246  ABC_Rad50
pfam1330475-245  AAA_21
cd03238187-246  ABC_UvrA
cd0328963-244  ABCC_CFTR2
cd03271134-244  ABC_UvrA_II
PRK1354060-244  PRK13540
cd03222181-242  ABC_RNaseL_inhibitor
cd0328834-222  ABCC_SUR2
cd03270187-245  ABC_UvrA_I
PRK1354178-246  PRK13541
pfam1347672-91  AAA_23
TIGR01247465-570  drrB
TIGR0095555-649  3a01204
PLN0321137-652  PLN03211
TIGR0095627-568  3a01205
TIGR0095651-652  3a01205
PLN0314062-573  PLN03140
COG113160-338  CcmA
PLN0314063-651  PLN03140
COG112060-274  FepC
COG455577-301  NatA
COG113660-246  LolD
COG112161-274  ZnuC
TIGR0118877-272  drrA
TIGR0360860-245  L_ocin_972_ABC
COG384261-294  PotA
COG111660-243  TauB
COG112760-274  MlaF
COG112255-274  EcfA2
COG363861-273  PhnC
TIGR0298260-264  heterocyst_DevA
COG383960-294  MalK
TIGR0386476-275  PQQ_ABC_ATP
TIGR0231553-272  ABC_phnC
COG414873-275  ModC
COG384077-275  ThiQ
TIGR0267362-246  FtsE
TIGR0337564-274  type_I_sec_LssB
COG498864-245  CydD
TIGR0214274-275  modC_ABC
TIGR0286856-245  CydC
COG227460-289  SunT
COG112360-274  GsiA
COG112477-272  DppF
COG452563-262  TauB
COG461963-273  FetA
COG498763-277  CydC
PRK1116063-274  PRK11160
COG418163-246  YbbA
COG111960-268  ModF
TIGR0352279-243  GldA_ABC_ATP
TIGR0325863-294  PhnT
TIGR0096864-295  3a0106s01
COG113577-272  AbcC
COG041062-274  LivF
TIGR0285758-245  CydD
COG112559-328  OpuBA
TIGR0221156-264  LolD_lipo_ex
PRK1353960-245  PRK13539
PRK1123160-274  fecE
TIGR0374055-243  galliderm_ABC
PRK1058463-246  PRK10584
COG113260-274  MdlB
TIGR0116677-243  cbiO
COG458679-269  COG4586
TIGR0128878-268  nodI
COG112336-240  GsiA
COG460460-272  CeuD
COG455961-274  COG4559
PRK1353678-272  PRK13536
PRK1363662-272  cbiO
TIGR0387363-274  F420-0_ABC_ATP
COG041164-274  LivG
TIGR0341164-239  urea_trans_UrtD
COG288461-243  FtsE
PRK1427260-272  PRK14272
TIGR0220358-288  MsbA_lipidA
PRK1363958-272  cbiO
TIGR0220464-272  MsbA_rel
COG112964-269  MglA
PRK1124861-262  tauB
PRK1353778-272  PRK13537
COG111877-272  CysA
TIGR0440678-275  LPS_export_lptB
PRK1057577-272  PRK10575
PRK1365261-272  cbiO
TIGR0127777-264  thiQ
COG413660-219  YnjD
COG415260-273  YhaQ
TIGR0184260-274  type_I_sec_PrtD
COG384564-263  YufO
PRK1162959-243  lolD
COG113447-279  TagH
PRK1114474-272  modC
TIGR0452158-272  ECF_ATPase_2
PRK1100080-243  PRK11000
COG113760-272  LptB
COG413378-246  CcmA
COG039661-284  SufC
COG461858-274  ArpD
TIGR0379658-272  NHLM_micro_ABC1
COG467464-268  COG4674
TIGR0125752-268  rim_protein
COG110157-230  PhnK
PRK1425061-243  PRK14250
TIGR0184637-274  type_I_sec_HlyB
PRK1077177-274  thiQ
PRK1354835-274  hmuV
TIGR0118778-264  potA
TIGR0125771-243  rim_protein
COG044463-272  DppD
COG112660-243  GlnQ
COG416178-270  ArtP
PRK1025377-272  PRK10253
PRK1365764-272  PRK13657
PRK1024760-273  PRK10247
TIGR0231464-272  ABC_MetN
PRK0953677-274  btuD
PRK1053562-245  PRK10535
PRK1363758-272  cbiO
COG048861-217  Uup
PRK0998477-272  PRK09984
PRK1353878-245  PRK13538
TIGR0118464-262  ntrCD
COG526559-264  ATM1
PRK1061960-280  PRK10619
TIGR0377175-243  anch_rpt_ABC
TIGR0118678-301  proV
TIGR0095860-244  3a01208
PRK0945261-243  potA
COG417260-272  YejF
PRK1513448-243  PRK15134
PRK1112478-244  artP
PRK1426260-272  PRK14262
TIGR0341578-272  ABC_choXWV_ATP
PRK0369578-274  PRK03695
COG417578-292  ProV
TIGR0326563-217  PhnT2
PRK1089578-274  PRK10895
PRK1365158-243  PRK13651
COG112978-240  MglA
PRK1078960-287  PRK10789
COG460836-272  AppF
TIGR0232459-245  CP_lyasePhnL
COG416777-274  SapF
TIGR0097260-272  3a0107s01c2
PRK1354763-274  hmuV
PRK1543962-272  PRK15439
PRK1126461-272  PRK11264
TIGR0371958-220  ABC_ABC_ChvD
COG417247-274  YejF
PRK1128864-264  araG
PRK1090861-243  PRK10908
COG413878-274  BtuD
TIGR0326961-277  met_CoM_red_A2
TIGR0197860-282  sufC
COG111760-243  PstB
COG459877-275  HisP
TIGR0276935-265  nickel_nikE
PRK0970064-262  PRK09700
TIGR0277077-272  nickel_nikD
CHL0013160-284  ycf16
PRK1364464-274  cbiO
PRK1364777-243  cbiO
PRK1424762-272  PRK14247
PRK1364158-272  cbiO
PRK1424564-243  PRK14245
PRK0949362-274  glnQ
COG477849-243  PhnL
PRK1423960-229  PRK14239
TIGR0341077-219  urea_trans_UrtE
TIGR0119277-272  chvA
PRK1427460-243  PRK14274
PRK1364658-243  cbiO
COG048860-217  Uup
PRK13638181-278  cbiO
PRK1117477-244  PRK11174
PRK1427161-272  PRK14271
TIGR0119362-279  bacteriocin_ABC
PRK1426762-272  PRK14267
PRK1170177-231  phnK
PRK15134187-271  PRK15134
PRK13631185-272  cbiO
PRK1424660-272  PRK14246
PLN0323246-272  PLN03232
PRK1041956-237  nikE
PRK1143263-303  fbpC
PRK1424962-272  PRK14249
COG384577-273  YufO
PRK1426960-282  PRK14269
PRK1425560-243  PRK14255
PRK1181958-217  PRK11819
PRK1160770-217  potG
PRK1363456-272  cbiO
TIGR0452060-242  ECF_ATPase_1
PRK1161478-266  livF
PRK1425675-243  PRK14256
PRK1364869-242  cbiO
TIGR0300577-280  ectoine_ehuA
PRK1424461-272  PRK14244
PRK1007078-295  PRK10070
PRK1085162-218  PRK10851
PRK1115378-244  metN
PRK1364358-243  cbiO
PRK1424177-273  PRK14241
PRK1426860-273  PRK14268
PRK1511277-240  PRK15112
PRK1425175-272  PRK14251
TIGR0232365-231  CP_lyasePhnK
PLN0313046-224  PLN03130
PRK1364958-243  cbiO
PRK1041877-272  nikD
PRK1074464-221  pstB
TIGR0095770-274  MRP_assoc_pro
PRK0958060-268  sufC
PRK1425264-243  PRK14252
COG417830-246  YddA
COG124578-219  Rli1
PRK1098264-263  PRK10982
PRK1340978-217  PRK13409
PRK1505677-271  PRK15056
PRK1426045-292  PRK14260
PRK1425360-292  PRK14253
PTZ0024359-268  PTZ00243
PRK1363258-274  cbiO
PRK1426160-239  PRK14261
PRK0954460-217  znuC
PRK1354964-263  PRK13549
PRK1364556-268  cbiO
PRK1165078-217  ugpC
PRK1427364-243  PRK14273
PRK1426660-243  PRK14266
COG410765-229  PhnK
PRK09473187-272  oppD
PRK1363577-242  cbiO
TIGR0263378-272  xylG
TIGR0127163-289  CFTR_protein
PRK0970080-264  PRK09700
PRK11147160-243  PRK11147
PRK1424060-243  PRK14240
PRK1424260-243  PRK14242
PRK1079060-274  PRK10790
PRK1364060-242  cbiO
PRK1130077-217  livG
TIGR0119478-265  cyc_pep_trnsptr
TIGR0379763-272  NHLM_micro_ABC2
COG4170189-274  SapD
TIGR0263364-244  xylG
PRK15439181-240  PRK15439
TIGR0326978-275  met_CoM_red_A2
PTZ0026556-220  PTZ00265
PTZ00265124-285  PTZ00265
PRK1427557-272  PRK14275
PRK1423660-221  PRK14236
PRK1128867-240  araG
PRK1426370-290  PRK14263
PRK1076262-239  PRK10762
PRK10261186-243  PRK10261
PRK1423777-243  PRK14237
PRK10982183-239  PRK10982
PRK1130877-228  dppF
COG0419154-239  SbcC
pfam12698427-571  ABC2_membrane_3
PRK1424860-272  PRK14248
PRK1425870-292  PRK14258
PRK1117660-274  PRK11176
COG124570-239  Rli1
TIGR00630178-239  uvra
PRK1426477-243  PRK14264
PRK13549103-240  PRK13549
COG0178128-239  UvrA
PRK1425761-241  PRK14257
PRK13409158-217  PRK13409
PRK15079187-290  PRK15079
PRK00635186-243  PRK00635
PRK1423860-243  PRK14238
TIGR0127161-244  CFTR_protein
PRK1354380-217  PRK13543
PRK1354547-243  tagH
PRK1425477-239  PRK14254
PRK1076277-262  PRK10762
PRK1424370-273  PRK14243
PRK1093877-239  PRK10938
COG0842385-572  YadH
PRK15093189-274  PRK15093
COG0842394-581  YadH
PRK1364260-242  cbiO
PRK00635186-274  PRK00635
PRK11022186-243  dppD
PLN03073187-243  PLN03073
PRK13633187-243  PRK13633
COG041945-91  SbcC
PRK1026136-243  PRK10261
TIGR03719187-223  ABC_ABC_ChvD


Ontology Information


   
HPRD ID19411
Molecular ClassTransport/cargo protein
Molecular FunctionMolecular function unknown (GO:0005554)
Biological ProcessBiological_process unknown (GO:0000004)  



SNP Information


View SNP Geneview Report   

Drug Information


Uniprot ID DrugBank ID Name Type
Q9UNQ0DB00091CyclosporineSmallMoleculeDrug
Q9UNQ0DB00158Folic AcidSmallMoleculeDrug
Q9UNQ0DB00175PravastatinSmallMoleculeDrug
Q9UNQ0DB00213PantoprazoleSmallMoleculeDrug
Q9UNQ0DB00220NelfinavirSmallMoleculeDrug
Q9UNQ0DB00242CladribineSmallMoleculeDrug
Q9UNQ0DB00255DiethylstilbestrolSmallMoleculeDrug
Q9UNQ0DB00285VenlafaxineSmallMoleculeDrug
Q9UNQ0DB00286Conjugated EstrogensSmallMoleculeDrug
Q9UNQ0DB00317GefitinibSmallMoleculeDrug
Q9UNQ0DB00338OmeprazoleSmallMoleculeDrug
Q9UNQ0DB00398SorafenibSmallMoleculeDrug
Q9UNQ0DB00444TeniposideSmallMoleculeDrug
Q9UNQ0DB00448LansoprazoleSmallMoleculeDrug
Q9UNQ0DB00457PrazosinSmallMoleculeDrug
Q9UNQ0DB00470DronabinolSmallMoleculeDrug
Q9UNQ0DB00495ZidovudineSmallMoleculeDrug
Q9UNQ0DB00503RitonavirSmallMoleculeDrug
Q9UNQ0DB00515CisplatinSmallMoleculeDrug
Q9UNQ0DB00526OxaliplatinSmallMoleculeDrug
Q9UNQ0DB00530ErlotinibSmallMoleculeDrug
Q9UNQ0DB00541VincristineSmallMoleculeDrug
Q9UNQ0DB00544FluorouracilSmallMoleculeDrug
Q9UNQ0DB00549ZafirlukastSmallMoleculeDrug
Q9UNQ0DB00563MethotrexateSmallMoleculeDrug
Q9UNQ0DB00602IvermectinSmallMoleculeDrug
Q9UNQ0DB00619ImatinibSmallMoleculeDrug
Q9UNQ0DB00624TestosteroneSmallMoleculeDrug
Q9UNQ0DB00631ClofarabineSmallMoleculeDrug
Q9UNQ0DB00655EstroneSmallMoleculeDrug
Q9UNQ0DB00661VerapamilSmallMoleculeDrug
Q9UNQ0DB00669SumatriptanSmallMoleculeDrug
Q9UNQ0DB00675TamoxifenSmallMoleculeDrug
Q9UNQ0DB00688Mycophenolate mofetilSmallMoleculeDrug
Q9UNQ0DB00694DaunorubicinSmallMoleculeDrug
Q9UNQ0DB00698NitrofurantoinSmallMoleculeDrug
Q9UNQ0DB00709LamivudineSmallMoleculeDrug
Q9UNQ0DB00740RiluzoleSmallMoleculeDrug
Q9UNQ0DB00741HydrocortisoneSmallMoleculeDrug
Q9UNQ0DB00762IrinotecanSmallMoleculeDrug
Q9UNQ0DB00773EtoposideSmallMoleculeDrug
Q9UNQ0DB00783EstradiolSmallMoleculeDrug
Q9UNQ0DB00795SulfasalazineSmallMoleculeDrug
Q9UNQ0DB00921BuprenorphineSmallMoleculeDrug
Q9UNQ0DB00958CarboplatinSmallMoleculeDrug
Q9UNQ0DB00966TelmisartanSmallMoleculeDrug
Q9UNQ0DB00970DactinomycinSmallMoleculeDrug
Q9UNQ0DB00973EzetimibeSmallMoleculeDrug
Q9UNQ0DB00997DoxorubicinSmallMoleculeDrug
Q9UNQ0DB01016GlyburideSmallMoleculeDrug
Q9UNQ0DB01030TopotecanSmallMoleculeDrug
Q9UNQ0DB01051NovobiocinSmallMoleculeDrug
Q9UNQ0DB01094HesperetinSmallMoleculeDrug
Q9UNQ0DB01097LeflunomideSmallMoleculeDrug
Q9UNQ0DB01098RosuvastatinSmallMoleculeDrug
Q9UNQ0DB01129RabeprazoleSmallMoleculeDrug
Q9UNQ0DB01204MitoxantroneSmallMoleculeDrug
Q9UNQ0DB01229PaclitaxelSmallMoleculeDrug
Q9UNQ0DB01232SaquinavirSmallMoleculeDrug
Q9UNQ0DB01234DexamethasoneSmallMoleculeDrug
Q9UNQ0DB01248DocetaxelSmallMoleculeDrug
Q9UNQ0DB01254DasatinibSmallMoleculeDrug
Q9UNQ0DB01268SunitinibSmallMoleculeDrug
Q9UNQ0DB04868NilotinibSmallMoleculeDrug
Q9UNQ0DB05239CobimetinibSmallMoleculeDrug
Q9UNQ0DB05294VandetanibSmallMoleculeDrug
Q9UNQ0DB06589PazopanibSmallMoleculeDrug
Q9UNQ0DB06605ApixabanSmallMoleculeDrug
Q9UNQ0DB06772CabazitaxelSmallMoleculeDrug
Q9UNQ0DB08828VismodegibSmallMoleculeDrug
Q9UNQ0DB08860PitavastatinSmallMoleculeDrug
Q9UNQ0DB08864RilpivirineSmallMoleculeDrug
Q9UNQ0DB08880TeriflunomideSmallMoleculeDrug
Q9UNQ0DB08881VemurafenibSmallMoleculeDrug
Q9UNQ0DB08896RegorafenibSmallMoleculeDrug
Q9UNQ0DB08901PonatinibSmallMoleculeDrug
Q9UNQ0DB08912DabrafenibSmallMoleculeDrug
Q9UNQ0DB08916AfatinibSmallMoleculeDrug
Q9UNQ0DB08934SofosbuvirSmallMoleculeDrug
Q9UNQ0DB09054IdelalisibSmallMoleculeDrug
Q9UNQ0DB09065CobicistatSmallMoleculeDrug
Q9UNQ0DB09078LenvatinibSmallMoleculeDrug
Q9UNQ0DB09102DaclatasvirSmallMoleculeDrug
Q9UNQ0DB09291RolapitantSmallMoleculeDrug
Q9UNQ0DB09330OsimertinibSmallMoleculeDrug
Q9UNQ0DB11363AlectinibSmallMoleculeDrug

External Links


                                 
ArrayExpressGO
ICGCGO
Cancer3DGO
COSMICGO
NCGGO
TSGeneGO
Tumor Gene Family of DatabasesGO
CCDBGO
G2SBCGO
Osteosarcoma DatabaseGO
RCDBGO